SCHEMBL9029970

SCHEMBL9029970

O=c1n(Cc2ccccc2)c2nc[nH]c2c2nnc(-c3ccncc3)n12

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.52
ADORA3 P0DMS8 1/20 0.49
ADORA2B P29275 1/20 0.49
PDE4A P27815 6/20 0.48
PDE4B Q07343 6/20 0.48
PDE4C Q08493 6/20 0.48
PDE4D Q08499 6/20 0.48
KMT2A Q03164 2/20 0.48
POLB P06746 2/20 0.47
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9030884 0.82 PNP (0.57) PNPADORA3ADORA2BPDE4APDE4B
SCHEMBL9029804 0.82 PDE4A (0.58) ADORA3ADORA2BPDE4APDE4BPDE4C
SCHEMBL9030966 0.80 PDE4A (0.55) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL9032044 0.78 PDE4A (0.56) ADORA3ADORA2BPDE4APDE4BPDE4C
SCHEMBL3107001 0.74 ADORA3 (0.78) PNPADORA3ADORA2BPDE4APDE4B
SCHEMBL9029959 0.72 PDE4A (0.54) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL9030681 0.71 HPGD (0.51) ADORA2BKMT2APOLBKDM4E
SCHEMBL9119046 0.71 ADORA2B (0.81) PNPADORA3ADORA2BPDE4APDE4B
SCHEMBL9030631 0.71 ADORA2B (0.46) ADORA2BPDE4APDE4BPDE4CPDE4D
SCHEMBL9032111 0.69 PNP (1.00) PNPADORA3ADORA2BPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0417790-B1 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-12-04 EP claimed
US-5173492-A Bronchodilator agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-12-22 US claimed
EP-0417790-B1 S-triazolo[3,4-i]purine derivatives KYOWA HAKKO KOGYO KK (JP) 1996-12-04 EP disclosed
US-5173492-A Bronchodilator agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-12-22 US disclosed