SCHEMBL903087

SCHEMBL903087

Cc1nnn(C)c1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
HCAR3 P49019 1/20 0.38
L3MBTL1 Q9Y468 3/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
POLB P06746 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
KDM4E B2RXH2 4/20 0.35
MEN1 O00255 1/20 0.35
PABPC1 P11940 1/20 0.35
KMT2A Q03164 1/20 0.35
GRIA1 P42261 2/20 0.33
GRIA2 P42262 2/20 0.33
GRIA3 P42263 2/20 0.33
GRIA4 P48058 2/20 0.33
PTGES O14684 2/20 0.33
GRN P28799 1/20 0.33
SORT1 Q99523 1/20 0.33
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16442926 0.80 MEN1 (0.41) HCAR3L3MBTL1ALDH1A1GAAKDM4E
SCHEMBL23656484 0.77 GRIA4 (0.44) NPC1HCAR3L3MBTL1MAPTPOLB
SCHEMBL9914070 0.77 NPC1 (0.57) NPC1HCAR3L3MBTL1MAPTPOLB
SCHEMBL903085 0.77 NPSR1 (0.37) NPC1L3MBTL1ALDH1A1GAAPOLB
SCHEMBL23362848 0.76 NPC1 (0.37) NPC1HCAR3L3MBTL1MAPTPOLB
SCHEMBL15897056 0.76 NPC1 (0.37) NPC1HCAR3L3MBTL1MAPTPOLB
SCHEMBL20614568 0.75 SMN1; SMN2 (0.41) ALDH1A1KDM4EKMT2ASMN1; SMN2
SCHEMBL14258066 0.74 NPC1 (0.44) NPC1HCAR3L3MBTL1MAPTPOLB
SCHEMBL4763456 0.73 MAPT (0.44) L3MBTL1MAPTALDH1A1GAAPOLB
SCHEMBL1889853 0.71 L3MBTL1 (0.43) NPC1L3MBTL1MAPTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2703406-A1 NOVEL CEPHEM COMPOUND HAVING CATECHOL OR PSEUDO-CATECHOL STRUCTURE Shionogi & Co., Ltd. (JP) 2014-03-05 EP disclosed
WO-2012044531-A1 NOVEL PIPERAZINE ANALOGS WITH SUBSTITUTED HETEROARYL GROUPS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-04-05 WO disclosed
WO-2012033736-A1 NOVEL PIPERAZINE ANALOGS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-15 WO disclosed