SCHEMBL903085

SCHEMBL903085

COC(=O)c1c(C)nnn1C

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
KDM4E B2RXH2 6/20 0.36
ALDH1A1 P00352 4/20 0.35
HTT P42858 1/20 0.35
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
GAA P10253 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
PABPC1 P11940 1/20 0.33
EIF4H Q15056 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PTGES O14684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9881658 0.81 KMT2A (0.46) NPSR1L3MBTL1KDM4EALDH1A1POLB
SCHEMBL1930001 0.80 ALDH1A1 (0.48) NPSR1ALDH1A1HTTGAAMEN1
SCHEMBL31667226 0.78 ALDH1A1 (0.40) NPSR1L3MBTL1KDM4EALDH1A1HTT
SCHEMBL903087 0.77 NPC1 (0.38) L3MBTL1KDM4EALDH1A1HTTNPC1
SCHEMBL729060 0.76 L3MBTL1 (0.46) NPSR1L3MBTL1KDM4EALDH1A1HTT
SCHEMBL1412412 0.76 NPC1 (0.47) NPSR1KDM4EALDH1A1NPC1GAA
SCHEMBL16442926 0.75 MEN1 (0.41) L3MBTL1KDM4EALDH1A1GAAMEN1
SCHEMBL9194890 0.74 KDM4E (0.42) NPSR1L3MBTL1KDM4EALDH1A1POLB
SCHEMBL25759724 0.74 SMN1; SMN2 (0.50) NPSR1L3MBTL1KDM4EALDH1A1NPC1
SCHEMBL1930172 0.73 NPSR1 (0.43) NPSR1KDM4EALDH1A1HTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044531-A1 NOVEL PIPERAZINE ANALOGS WITH SUBSTITUTED HETEROARYL GROUPS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-04-05 WO disclosed
US-20090209430-A1 TEMPLATE DIRECTED SPLIT AND MIX SYSTHESIS OF SMALL MOLECULE LIBRARIES NUEVOLUTION A/S (DK) 2009-08-20 US disclosed