SCHEMBL903134

SCHEMBL903134

COc1ccc2ccccc2c1-c1noc(C)c1C(=O)N1CCN(c2ccc([N+](=O)[O-])cc2Cl)CC1

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.57
MAPK1 P28482 2/20 0.55
ALDH1A1 P00352 7/20 0.51
KDM4E B2RXH2 3/20 0.51
GAA P10253 1/20 0.51
LMNA P02545 6/20 0.51
MAPT P10636 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
SLC6A5 Q9Y345 2/20 0.47
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
HTT P42858 2/20 0.45
POLB P06746 1/20 0.45
TP53 P04637 1/20 0.44
SLC6A9 P48067 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12691880 0.94 TSHR (0.59) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL10082091 0.86 TSHR (0.68) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL899837 0.83 TSHR (0.56) TSHRMAPK1ALDH1A1KDM4EGAA
Nucleozin SCHEMBL1225006 0.83 NPC1 (0.61) TSHRALDH1A1KDM4EGAALMNA
Nucleozin SCHEMBL29360670 0.83 NPC1 (0.61) TSHRALDH1A1KDM4EGAALMNA
SCHEMBL899570 0.82 LMNA (0.67) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL10082093 0.81 LMNA (0.57) TSHRMAPK1ALDH1A1KDM4ELMNA
SCHEMBL898748 0.81 LMNA (0.57) TSHRMAPK1ALDH1A1KDM4ELMNA
SCHEMBL12691812 0.81 ALDH1A1 (0.59) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL899632 0.81 LMNA (0.57) TSHRMAPK1ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2621920-B1 NOVEL PIPERAZINE ANALOGS WITH SUBSTITUTED HETEROARYL GROUPS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL MYERS SQUIBB CO (US) 2016-01-27 EP disclosed
WO-2012044531-A1 NOVEL PIPERAZINE ANALOGS WITH SUBSTITUTED HETEROARYL GROUPS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-04-05 WO disclosed