SCHEMBL9034360

SCHEMBL9034360

CC(=O)Nc1ccc2c(c1)CCC(C1C(=O)c3cc(NS(C)(=O)=O)ccc3OC13CCNCC3)C2

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.37
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
BAZ2B Q9UIF8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfuric Acid SCHEMBL9032305 0.88 KCNH2 (0.35) KCNH2
SCHEMBL7388072 0.87 KCNH2 (0.48) KCNH2
Hydrochloric Acid SCHEMBL7359212 0.86 KCNH2 (0.48) KCNH2
SCHEMBL9039225 0.81 KCNH2 (0.32) KCNH2
Hydrochloric Acid SCHEMBL9041198 0.74 KCNH2 (0.37) KCNH2
Hydrochloric Acid SCHEMBL8564106 0.74 ADRA1D (0.37) KCNH2
SCHEMBL9039873 0.73 KCNH2 (0.50) KCNH2
SCHEMBL8831682 0.72 KCNH2 (0.55) KCNH2
SCHEMBL3457612 0.71 ADRA1D (0.37) ALDH1A1
Hydrochloric Acid SCHEMBL8832193 0.71 KCNH2 (0.54) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683782-A4 SPIRO (2H-1-BENZOPYRAN-2, 4' PIPERIDINE) CLASS III ANTIARRHYTHMICS. MERCK & CO INC (US) 1996-03-27 EP disclosed
EP-0683782-A1 SPIRO (2H-1-BENZOPYRAN-2, 4' PIPERIDINE) CLASS III ANTIARRHYTHMICS MERCK & CO. INC. (US) 1995-11-29 EP disclosed
WO-1994018204-A1 SPIRO (2H-1-BENZOPYRAN-2, 4' PIPERIDINE) CLASS III ANTIARRHYTHMICS MERCK & CO., INC. (US) 1994-08-18 WO disclosed