SCHEMBL9034715

SCHEMBL9034715

O=C1CCn2c(-c3ccccc3)nc3cc(Cl)cc1c32

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.48
KDM4E B2RXH2 3/20 0.43
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HTR3A P46098 1/20 0.40
CYP1A2 P05177 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
GAA P10253 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
EGFR P00533 1/20 0.39
CYP1A1 P04798 2/20 0.38
CYP1B1 Q16678 2/20 0.38
KCNH2 Q12809 2/20 0.38
GRM2 Q14416 2/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9034743 0.81 TUBB4A (0.47) PARP1KDM4ELMNAHTTL3MBTL1
SCHEMBL6199833 0.81 PARP1 (0.66) PARP1HTR3AKCNH2GRM2
SCHEMBL9035061 0.81 PARP1 (0.42) PARP1KDM4ELMNAHTTL3MBTL1
SCHEMBL8824023 0.78 PARP1 (0.68) PARP1HTR3AKCNH2GRM2
SCHEMBL9035190 0.75 PARP1 (0.41) PARP1KDM4ELMNAHTR3ANPC1
SCHEMBL6514531 0.69 SMN1; SMN2 (0.32) PARP1SMN1; SMN2
SCHEMBL423080 0.68 PARP1 (0.56) PARP1HTR3AKCNH2GRM2
SCHEMBL9036526 0.68 PARP1 (0.41) PARP1KDM4EHTR3ACYP1A2NPC1
SCHEMBL15543213 0.66 KDM4E (0.55) KDM4ELMNAHTTL3MBTL1CYP1A2
SCHEMBL6829416 0.66 PARP1 (0.36) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0405442-B1 4,5-Dihydro-6H-imidazo[4,5,1-ij]quinolin-6-one-6-oxime-O-sulfonic acid derivatives MOCHIDA PHARM CO LTD (JP) 1996-09-04 EP disclosed
US-5151431-A Diuretics MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1992-09-29 US disclosed
EP-0405442-A1 4,5-Dihydro-6H-imidazo[4,5,1-ij]quinolin-6-one-6-oxime-O-sulfonic acid derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-01-02 EP disclosed