SCHEMBL9035190

SCHEMBL9035190

O=C1CCn2c(-c3ccccc3)nc3c(Cl)ccc1c32

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.41
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
GAA P10253 1/20 0.35
HTR3A P46098 1/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TSHR P16473 1/20 0.34
THRB P10828 2/20 0.33
LMNA P02545 1/20 0.33
PBRM1 Q86U86 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9034379 0.87 ALDH1A1 (0.37) PARP1NPC1MAPTRAB9AAPOBEC3G
SCHEMBL9035008 0.81 KDM4E (0.35) PARP1GAAALDH1A1HPGDKDM4E
SCHEMBL9035014 0.81 KDM4E (0.35) PARP1GAAALDH1A1HPGDKDM4E
SCHEMBL9035474 0.80 GRM5 (0.35) NPC1MAPTRAB9AALDH1A1HPGD
SCHEMBL6199833 0.77 PARP1 (0.66) PARP1HTR3AKCNH2GRM2
SCHEMBL9034715 0.75 PARP1 (0.48) PARP1NPC1RAB9AGAAHTR3A
SCHEMBL9035061 0.72 PARP1 (0.42) PARP1NPC1RAB9AGAAHTR3A
SCHEMBL8824023 0.71 PARP1 (0.68) PARP1HTR3AKCNH2GRM2
SCHEMBL9035248 0.71 LMNA (0.33) PARP1MAPTALDH1A1HPGDKDM4E
SCHEMBL6139581 0.71 PARP1 (0.32) PARP1MAPTGAAKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0405442-B1 4,5-Dihydro-6H-imidazo[4,5,1-ij]quinolin-6-one-6-oxime-O-sulfonic acid derivatives MOCHIDA PHARM CO LTD (JP) 1996-09-04 EP disclosed
US-5151431-A Diuretics MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1992-09-29 US disclosed
EP-0405442-A1 4,5-Dihydro-6H-imidazo[4,5,1-ij]quinolin-6-one-6-oxime-O-sulfonic acid derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-01-02 EP disclosed