SCHEMBL9034796

SCHEMBL9034796

COc1ccccc1N1CCN(CCNC(=O)c2nsc3ccccc23)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.65
ADRA1A P35348 2/20 0.65
DRD2 P14416 3/20 0.65
DRD4 P21917 1/20 0.65
HTR2A P28223 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9036734 0.99 HTR1A (0.64) HTR1AADRA1ADRD2DRD4HTR2A
SCHEMBL9467179 0.94 DRD2 (0.69) HTR1ADRD2DRD4HTR2A
Hydrochloric Acid SCHEMBL9035124 0.94 DRD2 (0.68) HTR1ADRD2DRD4HTR2A
SCHEMBL9474121 0.94 DRD2 (0.73) HTR1AADRA1ADRD2DRD4HTR2A
Hydrochloric Acid SCHEMBL9037059 0.93 DRD2 (0.72) HTR1AADRA1ADRD2DRD4HTR2A
SCHEMBL9466381 0.87 DRD2 (0.52) HTR1AADRA1ADRD2DRD4HTR2A
Hydrochloric Acid SCHEMBL9035828 0.86 DRD2 (0.51) HTR1AADRA1ADRD2DRD4HTR2A
SCHEMBL9466203 0.85 DRD3 (0.66) HTR1ADRD2DRD4HTR2A
SCHEMBL9036875 0.85 DRD3 (0.66) HTR1ADRD2DRD4HTR2A
SCHEMBL9036862 0.85 DRD3 (0.66) HTR1ADRD2DRD4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5225412-A Antipsychotic HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-06 US claimed
EP-0511610-B1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST ROUSSEL PHARMA (US) 1996-09-11 EP disclosed
US-5225412-A Antipsychotic HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-06 US disclosed
EP-0511610-A1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-11-04 EP disclosed
US-5143923-A Psychological disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-09-01 US disclosed