SCHEMBL9034922

SCHEMBL9034922

C1CN(Cc2nn[nH]c2CN2CCOCC2)CCO1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TYMP P19971 1/20 0.41
CXCR4 P61073 1/20 0.40
PARP1 P09874 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP2C9 P11712 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HPGD P15428 1/20 0.36
CYP2A13 Q16696 5/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LMNA P02545 1/20 0.35
THRB P10828 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTPN1 P18031 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9035977 0.92 HRH3 (0.38) TYMPCXCR4PARP1HRH3ALDH1A1
SCHEMBL1610726 0.90 NCF1 (0.41) TYMPCXCR4PARP1HRH3ALDH1A1
SCHEMBL12715997 0.88 CXCR4 (0.37) TYMPCXCR4PARP1HRH3ALDH1A1
SCHEMBL18377716 0.81 CYP2A13 (0.40) TYMPCXCR4HRH3ALDH1A1CYP2C9
SCHEMBL19589388 0.77 ALOX15 (0.45) TYMPCXCR4HRH3ALDH1A1CYP2C9
SCHEMBL9034911 0.77 HTR1D (0.38) TYMPPARP1
SCHEMBL4982004 0.69 HPGD (0.43) CXCR4HRH3ALDH1A1CYP2C9ALOX15
SCHEMBL19634969 0.66 PARP1 (0.37) TYMPCXCR4PARP1HRH3ALDH1A1
SCHEMBL2648324 0.64 ALDH1A1 (0.41) CXCR4HRH3ALDH1A1CYP2C9ALOX15
SCHEMBL2648327 0.64 CXCR4 (0.51) CXCR4HRH3ALDH1A1CYP2C9ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737192-A1 SUBSTITUTED MORPHOLINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 1996-10-16 EP disclosed
WO-1995018124-A1 SUBSTITUTED MORPHOLINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 1995-07-06 WO disclosed