SCHEMBL9036385

SCHEMBL9036385

COc1cc2c3c(c1)nc(-c1ccccc1)n3CC/C2=N\O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.38
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
PDE5A O76074 2/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
CYP1A1 P04798 4/20 0.35
CYP1A2 P05177 4/20 0.35
CYP1B1 Q16678 4/20 0.35
NPC1 O15118 1/20 0.35
ESR1 P03372 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
NFKB1 P19838 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
KMT2A Q03164 1/20 0.35
RELA Q04206 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9036389 1.00 PARP1 (0.38) PARP1KDM4EALDH1A1HPGDPDE5A
SCHEMBL9036526 0.84 PARP1 (0.41) PARP1KDM4EPDE5ACYP1A1CYP1A2
SCHEMBL9034743 0.83 TUBB4A (0.47) PARP1KDM4EALDH1A1HPGDPDE5A
SCHEMBL9243355 0.80 PARP1 (0.55) PARP1KDM4EHPGDRECQL
SCHEMBL8824093 0.80 PARP1 (0.55) PARP1KDM4EHPGDRECQL
SCHEMBL8824032 0.73 PARP1 (0.42) PARP1KDM4ERECQL
SCHEMBL8824037 0.73 PARP1 (0.42) PARP1KDM4ERECQL
SCHEMBL8823994 0.70 PARP1 (0.58) PARP1KDM4ENPC1RAB9AKMT2A
SCHEMBL9035014 0.70 KDM4E (0.35) PARP1KDM4EALDH1A1HPGDCYP1A2
SCHEMBL9035008 0.70 KDM4E (0.35) PARP1KDM4EALDH1A1HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0405442-B1 4,5-Dihydro-6H-imidazo[4,5,1-ij]quinolin-6-one-6-oxime-O-sulfonic acid derivatives MOCHIDA PHARM CO LTD (JP) 1996-09-04 EP disclosed
US-5151431-A Diuretics MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1992-09-29 US disclosed
EP-0405442-A1 4,5-Dihydro-6H-imidazo[4,5,1-ij]quinolin-6-one-6-oxime-O-sulfonic acid derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-01-02 EP disclosed