SCHEMBL903657

SCHEMBL903657

C[Si](C)(C)CCOCn1c([C@@H]2CCCN2)cnc1Br

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 2/20 0.33
CREBBP Q92793 1/20 0.31
CHRM2 P08172 3/20 0.30
CHRM4 P08173 2/20 0.30
CHRM5 P08912 2/20 0.30
CHRM1 P11229 2/20 0.30
CHRM3 P20309 2/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNA7 P36544 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30204428 0.79
SCHEMBL30204358 0.75 PRPS1 (0.33)
SCHEMBL15572246 0.73 DGAT1 (0.40) DGAT1
SCHEMBL15368135 0.73 DGAT1 (0.40) DGAT1
SCHEMBL15471725 0.72 DGAT1 (0.41) DGAT1
Hydrochloric Acid SCHEMBL535924 0.71 L3MBTL1 (0.34) DGAT1CHRM2CHRM4CHRM5CHRM1
SCHEMBL13070718 0.71 TAAR1 (0.33) DGAT1
SCHEMBL16105981 0.69 TAAR1 (0.36) DGAT1CHRM2CHRM4CHRM5CHRM1
SCHEMBL16105980 0.69 TAAR1 (0.36) DGAT1CHRM2CHRM4CHRM5CHRM1
SCHEMBL30889433 0.69 DGAT1 (0.37) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041014-A1 TETRACYCLIC INDOLE DERIVATIVES FOR TREATING HEPATITIS C VIRUS INFECTION MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed
WO-2011112429-A1 FUSED TRICYCLIC SILYL COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES SCHERING CORPORATION (US) 2011-09-15 WO disclosed