SCHEMBL9036613

SCHEMBL9036613

Cc1nc(N)nc(Cl)c1CCCCc1ccc(C(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.49
RARB P10826 6/20 0.49
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 1/20 0.48
RARA P10276 1/20 0.48
MAPT P10636 1/20 0.48
MTOR P42345 1/20 0.48
KMT2A Q03164 1/20 0.48
SCNN1A P37088 1/20 0.47
DHFR P00374 1/20 0.46
P2RX3 P56373 1/20 0.45
TLR8 Q9NR97 2/20 0.44
TLR7 Q9NYK1 2/20 0.44
POLB P06746 1/20 0.44
HPGD P15428 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CYP2D6 P10635 1/20 0.44
NPC1 O15118 1/20 0.44
NFKB1 P19838 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037084 0.89 CYP2D6 (0.55) RARBALDH1A1MEN1RARAMAPT
SCHEMBL9038207 0.86 DHFR (0.52) RARBALDH1A1MEN1RARAMAPT
SCHEMBL9338914 0.79 CYP2D6 (0.56) RARBALDH1A1MEN1RARAMAPT
SCHEMBL9343568 0.78 CYP2D6 (0.55) RARBALDH1A1MEN1RARAMAPT
SCHEMBL9215453 0.77 GART (0.52) NPSR1RARBALDH1A1MEN1RARA
SCHEMBL9341089 0.76 CYP2D6 (0.53) RARBALDH1A1MEN1RARAMAPT
SCHEMBL371605 0.74 RARB (0.71) RARBALDH1A1MEN1RARAMAPT
SCHEMBL9472454 0.73 RARB (0.72) RARBALDH1A1MEN1RARAMAPT
SCHEMBL30053056 0.73 RARB (0.72) RARBALDH1A1MEN1RARAMAPT
SCHEMBL15583704 0.73 RARB (0.72) RARBALDH1A1MEN1RARAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722440-A1 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES ELI LILLY AND COMPANY (US) 1996-07-24 EP disclosed
EP-0722440-A4 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES LILLY CO ELI (US) 1996-06-04 EP disclosed
US-5426110-A Inhibiting dihydrofolate reductase in mammals and treating susceptible reoplasms ELI LILLY AND COMPANY (US) 1995-06-20 US disclosed
WO-1995009845-A1 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES ELI LILLY AND COMPANY (US) 1995-04-13 WO disclosed