SCHEMBL9038207

SCHEMBL9038207

Nc1nc(N)c(CCCc2ccc(C(=O)O)cc2)c(Cl)n1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.52
CYP2D6 P10635 1/20 0.51
SCNN1A P37088 1/20 0.47
MAPT P10636 2/20 0.43
KMT2A Q03164 2/20 0.43
POLB P06746 1/20 0.43
ATM Q13315 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
RARB P10826 6/20 0.43
MBOAT4 Q96T53 1/20 0.42
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RARA P10276 1/20 0.41
MTOR P42345 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037084 0.97 CYP2D6 (0.55) DHFRCYP2D6SCNN1AMAPTKMT2A
SCHEMBL9341089 0.87 CYP2D6 (0.53) DHFRCYP2D6MAPTKMT2APOLB
SCHEMBL9036613 0.86 NPSR1 (0.49) DHFRCYP2D6SCNN1AMAPTKMT2A
SCHEMBL9338914 0.84 CYP2D6 (0.56) DHFRCYP2D6SCNN1AMAPTKMT2A
SCHEMBL9343568 0.83 CYP2D6 (0.55) DHFRCYP2D6SCNN1AMAPTKMT2A
SCHEMBL9037916 0.78 DHFR (0.69) DHFR
SCHEMBL9039506 0.75 DHFR (0.51) DHFR
SCHEMBL133470 0.74 RARB (0.68) MAPTKMT2ARARBMEN1ALDH1A1
SCHEMBL9339199 0.74 DHFR (0.54) DHFRCYP2D6SCNN1AMAPTKMT2A
SCHEMBL19143887 0.73 RARB (0.58) MAPTKMT2ARARBMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722440-A1 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES ELI LILLY AND COMPANY (US) 1996-07-24 EP disclosed
EP-0722440-A4 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES LILLY CO ELI (US) 1996-06-04 EP disclosed
US-5426110-A Inhibiting dihydrofolate reductase in mammals and treating susceptible reoplasms ELI LILLY AND COMPANY (US) 1995-06-20 US disclosed
WO-1995009845-A1 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES ELI LILLY AND COMPANY (US) 1995-04-13 WO disclosed