SCHEMBL9037181

SCHEMBL9037181

COc1ccc2[nH]cc(C(=O)N(C)CCCCN(C)c3ncccc3NC(C)C)c2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.45
NR4A2 P43354 1/20 0.43
CPT1A P50416 1/20 0.43
HTR2C P28335 1/20 0.43
LMNA P02545 4/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 2/20 0.42
MITF O75030 1/20 0.42
RAB9A P51151 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP2C9 P11712 1/20 0.41
IMPDH2 P12268 1/20 0.40
IMPDH1 P20839 1/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038042 0.95 KDR (0.46) KDRNR4A2CPT1AHTR2CLMNA
SCHEMBL9037383 0.87 HTR2C (0.41) KDRHTR2CLMNAKMT2AALDH1A1
SCHEMBL9038031 0.86 HTR2C (0.41) KDRHTR2CLMNACDK4CCND1
SCHEMBL9036372 0.85 HTR2C (0.41) KDRHTR2CLMNAKMT2AALDH1A1
SCHEMBL9242994 0.84 KMT2A (0.47) KDRNR4A2CPT1AHTR2CLMNA
SCHEMBL9037640 0.83 KDR (0.43) KDRKMT2AALDH1A1MTNR1AMTNR1B
SCHEMBL9038237 0.82 CDK4 (0.41) KDRHTR2CLMNAKMT2AALDH1A1
SCHEMBL9690016 0.79 KMT2A (0.48) KDRNR4A2CPT1AHTR2CLMNA
SCHEMBL8985813 0.77 CPT1A (0.45) KDRNR4A2CPT1AHTR2CLMNA
SCHEMBL9038843 0.74 LMNA (0.39) KDRNR4A2HTR2CLMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507861-B1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS UPJOHN CO (US) 1996-09-11 EP claimed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO claimed