SCHEMBL9036372

SCHEMBL9036372

CC(C)Nc1cccnc1N(C)CCCN(C)C(=O)c1c[nH]c2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.41
CDK4 P11802 11/20 0.40
CCND1 P24385 11/20 0.40
LMNA P02545 1/20 0.40
CDK2 P24941 2/20 0.39
KDR P35968 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037383 0.98 HTR2C (0.41) HTR2CCDK4CCND1LMNACDK2
SCHEMBL9038031 0.97 HTR2C (0.41) HTR2CCDK4CCND1LMNACDK2
SCHEMBL9038237 0.94 CDK4 (0.41) HTR2CCDK4CCND1LMNACDK2
SCHEMBL9038843 0.85 LMNA (0.39) HTR2CCDK4CCND1LMNACDK2
SCHEMBL9037181 0.85 KDR (0.45) HTR2CCDK4CCND1LMNAKDR
SCHEMBL9037640 0.83 KDR (0.43) CDK4CCND1KDRALDH1A1KMT2A
SCHEMBL9036635 0.82 CDK4 (0.43) HTR2CCDK4CCND1LMNACDK2
SCHEMBL9037086 0.82 CDK4 (0.42) HTR2CCDK4CCND1LMNACDK2
SCHEMBL9038042 0.81 KDR (0.46) HTR2CCDK4CCND1LMNAKDR
SCHEMBL9687990 0.80 HTR2C (0.43) HTR2CCDK4CCND1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507861-B1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS UPJOHN CO (US) 1996-09-11 EP claimed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO claimed