SCHEMBL9037640

SCHEMBL9037640

CC(C)Nc1cccnc1N(C)CCN(C)C(=O)c1c[nH]c2ccc(F)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.43
CDK4 P11802 4/20 0.38
CCND1 P24385 4/20 0.38
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
JAK2 O60674 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MPO P05164 2/20 0.35
CLK1 P49759 1/20 0.35
DYRK1A Q13627 1/20 0.35
DPP4 P27487 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
NOTUM Q6P988 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038237 0.88 CDK4 (0.41) KDRCDK4CCND1ALDH1A1KMT2A
SCHEMBL9038042 0.88 KDR (0.46) KDRCDK4CCND1MTNR1AMTNR1B
SCHEMBL9037181 0.83 KDR (0.45) KDRCDK4CCND1MTNR1AMTNR1B
SCHEMBL9037383 0.83 HTR2C (0.41) KDRCDK4CCND1ALDH1A1KMT2A
SCHEMBL9036372 0.83 HTR2C (0.41) KDRCDK4CCND1ALDH1A1KMT2A
SCHEMBL9689717 0.83 CDK4 (0.40) KDRCDK4CCND1KDM4EMPO
SCHEMBL9038031 0.82 HTR2C (0.41) KDRCDK4CCND1
SCHEMBL8985769 0.81 CDK4 (0.39) KDRCDK4CCND1POLBTDP1
SCHEMBL9038843 0.76 LMNA (0.39) KDRCDK4CCND1POLBGAA
SCHEMBL9037086 0.76 CDK4 (0.42) KDRCDK4CCND1POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507861-B1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS UPJOHN CO (US) 1996-09-11 EP claimed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO claimed