SCHEMBL903776

SCHEMBL903776

COc1ccc(F)c(C(Br)Br)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.41
ADRA2A P08913 2/20 0.40
ADRA1A P35348 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
GFER P55789 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
CA14 Q9ULX7 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17115832 0.83 CYP2D6 (0.43) CYP2D6ADRA2AADRA1ACHRM2CHRM1
SCHEMBL7937557 0.82 CYP2D6 (0.46) CYP2D6ADRA2AADRA1ACHRM2CHRM1
SCHEMBL11143567 0.81 CYP2D6 (0.44) CYP2D6ADRA2AADRA1AMEN1KMT2A
SCHEMBL2701413 0.80 CYP2D6 (0.41) CYP2D6ADRA2AADRA1ACHRM2CHRM1
SCHEMBL20256745 0.80 ADRA2A (0.46) CYP2D6ADRA2AADRA1ACHRM2CHRM1
SCHEMBL16960809 0.78 CYP2D6 (0.43) CYP2D6ADRA2AADRA1ACHRM2CHRM1
SCHEMBL31119047 0.78 ADRA2A (0.49) CYP2D6ADRA2AADRA1AMEN1KMT2A
SCHEMBL2823287 0.78 CYP2D6 (0.53) CYP2D6ADRA2AADRA1ACHRM2CHRM1
SCHEMBL3702003 0.78 CYP2D6 (0.53) CYP2D6ADRA2AADRA1ACHRM2CHRM1
SCHEMBL31119095 0.78 CYP2D6 (0.43) CYP2D6ADRA2AADRA1ACHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041014-A1 TETRACYCLIC INDOLE DERIVATIVES FOR TREATING HEPATITIS C VIRUS INFECTION MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed
US-7115766-B2 Nucleophilic approach for preparing radiolabeled imaging agents and associated compounds INDIANA UNIVERSITY RESEARCH & TECHNOLOGY CORP. (US) 2006-10-03 US disclosed
US-20040034246-A1 Nucleophilic approach for preparing radiolabeled imaging agents and associated compounds NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2004-02-19 US disclosed
WO-2002044144-A2 NUCLEOPHILIC APPROACH FOR PREPARING RADIOLABELED IMAGING AGENTS AND ASSOCIATED COMPOUNDS ADVANCED RESEARCH AND TECHNOLOGY INSTITUTE, INC. (US) 2002-06-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040034246-A1 Nucleophilic approach for preparing radiolabeled imaging agents and associated compounds SNCA, PARK7, SAMHD1 CYP2D6 3449/4885ADRA2A 2471/4885ADRA1A 2354/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.