SCHEMBL9038703

SCHEMBL9038703

O=[N+]([O-])c1cnc2c(c1)cc1c3c(cccc32)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.51
CYP3A4 P08684 1/20 0.51
ALOX15 P16050 1/20 0.51
HSD17B10 Q99714 1/20 0.51
MAPT P10636 6/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
TDP1 Q9NUW8 3/20 0.46
USP2 O75604 1/20 0.41
HPGD P15428 4/20 0.40
TSHR P16473 1/20 0.39
RECQL P46063 1/20 0.38
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214353 0.88 ALDH1A1 (0.41) ALDH1A1CYP3A4ALOX15HSD17B10MAPT
SCHEMBL9214349 0.85 MAPT (0.40) ALDH1A1CYP3A4ALOX15HSD17B10MAPT
SCHEMBL18573116 0.76 KDM4E (0.40) ALDH1A1CYP3A4ALOX15HSD17B10MAPT
SCHEMBL9078671 0.74 TYMS (0.43) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL9040658 0.73 MEN1 (0.66) ALDH1A1CYP3A4ALOX15HSD17B10MAPT
SCHEMBL9078669 0.72 MAPT (0.40) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL5376486 0.72 TDP1 (0.49) ALDH1A1CYP3A4ALOX15HSD17B10MAPT
SCHEMBL18573105 0.70 KDM4E (0.39) ALDH1A1HSD17B10MAPTMEN1KMT2A
SCHEMBL1074921 0.69 ALDH1A1 (0.59) ALDH1A1CYP3A4ALOX15MAPTMEN1
SCHEMBL30492617 0.69 ALDH1A1 (0.59) ALDH1A1CYP3A4ALOX15MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585382-A ANTICARCINOGENIC AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-17 US disclosed
EP-0705250-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-04-10 EP disclosed
US-5416089-A Antitumor agent THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-05-16 US disclosed
WO-1995000490-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-01-05 WO disclosed