SCHEMBL9078671

SCHEMBL9078671

O=C1OC(=O)c2cc3cc([N+](=O)[O-])cnc3c3cccc1c23

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 10/20 0.43
ALDH1A1 P00352 3/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MAPT P10636 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
S1PR4 O95977 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
XBP1 P17861 1/20 0.36
S1PR1 P21453 1/20 0.36
CCR6 P51684 1/20 0.36
AGTR1 P30556 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214353 0.90 ALDH1A1 (0.41) TYMSALDH1A1MEN1KMT2ATDP1
SCHEMBL9219065 0.81 MAPT (0.48) TYMSALDH1A1MEN1KMT2ATDP1
SCHEMBL9078930 0.79 CCR1 (0.45) TYMSMEN1KMT2AMAPTKDM4E
SCHEMBL9077614 0.78 ALDH1A1 (0.54) TYMSALDH1A1TSHR
SCHEMBL9077278 0.77 ALDH1A1 (0.40) TYMSALDH1A1MEN1KMT2ATSHR
SCHEMBL9079255 0.75 TYMS (0.47) TYMSALDH1A1MEN1KMT2ATSHR
SCHEMBL9038703 0.74 ALDH1A1 (0.51) ALDH1A1MEN1KMT2ATSHRTDP1
SCHEMBL9078696 0.74 TYMS (0.51) TYMSALDH1A1TSHRTDP1MAPT
SCHEMBL9208484 0.74 ALDH1A1 (0.41) TYMSALDH1A1MEN1KMT2ATDP1
SCHEMBL9209268 0.74 FTO (0.48) ALDH1A1MEN1KMT2ATDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585382-A ANTICARCINOGENIC AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-17 US disclosed
CN-1125943-A Diimide polycyclic and heterocyclic chromophores as antitumor agents DU PONT MERCK PHARMA (US) 1996-07-03 CN disclosed
US-5416089-A Antitumor agent THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-05-16 US disclosed
WO-1995000490-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-01-05 WO disclosed