SCHEMBL903904

SCHEMBL903904

c1cc(-n2cnnn2)ccc1OCCC1CC2(CCNCC2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.44
TDP1 Q9NUW8 2/20 0.44
BLM P54132 1/20 0.44
ALDH1A1 P00352 3/20 0.43
PKM P14618 1/20 0.43
MAPT P10636 2/20 0.42
KMT2A Q03164 4/20 0.42
MEN1 O00255 2/20 0.39
ALOX15 P16050 1/20 0.39
GPR119 Q8TDV5 1/20 0.39
CYP3A4 P08684 1/20 0.38
USP2 O75604 1/20 0.38
MAPK1 P28482 1/20 0.38
ATF4 P18848 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
ATM Q13315 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CTDSP1 Q9GZU7 1/20 0.36
F2 P00734 1/20 0.36
NOTUM Q6P988 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL904207 0.78 GPR119 (0.60) POLBTDP1BLMALDH1A1PKM
SCHEMBL904063 0.78 GPR119 (0.66) ALDH1A1PKMGPR119
SCHEMBL15486250 0.75 GPR119 (0.49) POLBTDP1BLMALDH1A1PKM
SCHEMBL12987784 0.75 GPR119 (0.49) POLBTDP1BLMALDH1A1PKM
SCHEMBL13195458 0.72 POLB (0.44) POLBTDP1BLMALDH1A1PKM
SCHEMBL4202083 0.70 CYP19A1 (0.63) POLBTDP1BLMALDH1A1PKM
SCHEMBL4207158 0.70 POLB (0.60) POLBTDP1BLMALDH1A1PKM
Hydrochloric Acid SCHEMBL13735667 0.68 TDP1 (0.44) POLBTDP1BLMALDH1A1PKM
Hydrochloric Acid SCHEMBL13735668 0.68 TDP1 (0.44) POLBTDP1BLMALDH1A1PKM
SCHEMBL8381009 0.68 NOTUM (0.51) POLBTDP1BLMALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed