SCHEMBL903956

SCHEMBL903956

CS(=O)(=O)c1ccc(-c2c(F)cc(O)cc2F)cc1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.53
PTGS2 P35354 16/20 0.53
KIF11 P52732 1/20 0.49
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL384337 0.79 PTGS2 (0.58) ENPP2PTGS2ESR1ESR2
SCHEMBL903934 0.76 KIF11 (0.58) ENPP2PTGS2KIF11
SCHEMBL28374796 0.76 ESR1 (0.67) KIF11ESR1ESR2
SCHEMBL16982125 0.76 ESR1 (0.67) KIF11ESR1ESR2
SCHEMBL386673 0.75 KIF11 (0.61) ENPP2PTGS2KIF11ESR1ESR2
SCHEMBL17775110 0.75 ESR1 (0.55) PTGS2ESR1ESR2
SCHEMBL16582458 0.74 ESR1 (0.59) ESR1ESR2
SCHEMBL388018 0.74 ENPP2 (0.86) ENPP2PTGS2ESR1ESR2
SCHEMBL30604305 0.72 PTGS2 (0.60) PTGS2
SCHEMBL386705 0.72 ENPP2 (0.55) ENPP2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102639500-A Tricyclic compound, preparation method and pharmaceutical use thereof SHANGHAI HENGRUI PHARM CO LTD 2012-08-15 CN disclosed
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed