SCHEMBL9039595

SCHEMBL9039595

CCOC(=O)c1ccc(OCCc2c[nH]c3nc(N)nc(N)c23)cc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.52
NAMPT P43490 1/20 0.44
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
RAB9A P51151 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7843188 0.86 NAMPT (0.57) DHFRNAMPTLMNA
SCHEMBL9042512 0.85 NAMPT (0.43) DHFRNAMPTLMNARAB9A
SCHEMBL9044536 0.84 NAMPT (0.51) DHFRNAMPTLMNA
SCHEMBL9040527 0.82 DHFR (0.51) DHFRL3MBTL1HSD17B10
SCHEMBL9040512 0.82 DHFR (0.51) DHFRL3MBTL1HSD17B10
SCHEMBL9040305 0.82 NAMPT (0.42) DHFRNAMPTLMNA
SCHEMBL9039740 0.81 DHFR (0.51) DHFRTDP1L3MBTL1NPC1LMNA
SCHEMBL9044792 0.77 TYMS (0.51) DHFRNAMPTNPC1LMNARAB9A
SCHEMBL9042706 0.76 DHFR (0.66) DHFR
SCHEMBL9047680 0.76 DHFR (0.45) DHFRNAMPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0400562-B1 Pyrrolopyrimidines, their production and use as tumoricidal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-08-21 EP disclosed