SCHEMBL9039740

SCHEMBL9039740

CCOC(=O)c1ccc(OCCc2c(O)[nH]c3nc(N)nc(N)c23)cc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.51
LMNA P02545 3/20 0.44
HSD17B10 Q99714 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAPT P10636 3/20 0.41
TBXAS1 P24557 1/20 0.40
ALDH1A1 P00352 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAOA P21397 1/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
TP53 P04637 1/20 0.39
STS P08842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9042572 0.84 MAPT (0.43) DHFRLMNAHSD17B10NPC1RAB9A
SCHEMBL9039595 0.81 DHFR (0.52) DHFRLMNAHSD17B10NPC1RAB9A
SCHEMBL8997197 0.74 DHFR (0.37) DHFR
SCHEMBL9794864 0.72 GART (0.59) DHFRLMNAHSD17B10NPC1RAB9A
SCHEMBL6701399 0.69 TDP1 (0.74) LMNAHSD17B10RAB9ATDP1L3MBTL1
SCHEMBL7843188 0.69 NAMPT (0.57) DHFRLMNACYP1A2CYP3A4MAOA
SCHEMBL9042512 0.68 NAMPT (0.43) DHFRLMNARAB9ACYP1A2CYP3A4
SCHEMBL9044536 0.67 NAMPT (0.51) DHFRLMNACYP1A2CYP3A4MAOA
SCHEMBL4247628 0.67 TDP1 (0.62) LMNATDP1L3MBTL1MAPTTBXAS1
SCHEMBL950916 0.67 L3MBTL1 (0.66) LMNATDP1L3MBTL1MAPTTBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0400562-B1 Pyrrolopyrimidines, their production and use as tumoricidal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-08-21 EP disclosed
EP-0400562-A1 Pyrrolopyrimidines, their production and use as tumoricidal agents Takeda Chemical Industries, Ltd. (JP) 1990-12-05 EP disclosed