SCHEMBL9039787

SCHEMBL9039787

O=C(O)c1cc2ccc(C(F)(F)F)cc2c2cccc(C(=O)OC(=O)c3cccc4c3c(C(=O)O)cc3ccc(C(F)(F)F)cc34)c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPL P40238 1/20 0.42
ALDH1A1 P00352 4/20 0.40
HPGD P15428 3/20 0.40
KDM4E B2RXH2 2/20 0.40
HSD17B10 Q99714 2/20 0.40
USP2 O75604 1/20 0.39
CYP2C19 P33261 1/20 0.39
MRGPRX4 Q96LA9 4/20 0.39
TAS2R14 Q9NYV8 2/20 0.38
GRIK1 P39086 3/20 0.38
SORT1 Q99523 3/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
CYP1A2 P05177 2/20 0.37
ALOX12 P18054 1/20 0.37
GAA P10253 1/20 0.37
GMNN O75496 1/20 0.37
LMNA P02545 1/20 0.37
TTR P02766 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9078976 0.83 KDM4E (0.40) ALDH1A1HPGDKDM4EHSD17B10MEN1
SCHEMBL9041814 0.81 NR4A1 (0.51) ALDH1A1HPGDKDM4EHSD17B10CYP2C19
SCHEMBL9080057 0.81 ALDH1A1 (0.41) MPLALDH1A1HPGDKDM4EHSD17B10
SCHEMBL9077953 0.79 CNR2 (0.40) ALDH1A1HPGDKDM4EHSD17B10CYP2C19
SCHEMBL9077610 0.78 ALDH1A1 (0.44) ALDH1A1HPGDMEN1KMT2ACYP3A4
SCHEMBL9079543 0.78 XDH (0.41) ALDH1A1HPGDKDM4EHSD17B10MCL1
SCHEMBL9079015 0.74 KDM4E (0.51) ALDH1A1HPGDKDM4EHSD17B10MEN1
SCHEMBL9078240 0.74 KDM4E (0.50) ALDH1A1HPGDKDM4EHSD17B10MEN1
SCHEMBL9217742 0.73 NR4A1 (0.43) ALDH1A1HPGDKDM4EHSD17B10MEN1
SCHEMBL9041045 0.72 CLK1 (0.42) ALDH1A1KDM4EMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585382-A ANTICARCINOGENIC AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-17 US disclosed
EP-0705250-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-04-10 EP disclosed
US-5416089-A Antitumor agent THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-05-16 US disclosed
WO-1995000490-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-01-05 WO disclosed