SCHEMBL9078976

SCHEMBL9078976

O=C(O)c1cc2ccc(F)cc2c2cccc(C(=O)OC(=O)c3cccc4c3c(C(=O)O)cc3ccc(F)cc34)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
DHODH Q02127 3/20 0.39
NR4A1 P22736 1/20 0.38
NR4A2 P43354 1/20 0.38
NR4A3 Q92570 1/20 0.38
GRIN2D O15399 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37
GRIN2C Q14957 1/20 0.37
PTPN1 P18031 1/20 0.37
PARP1 P09874 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36
KEAP1 Q14145 1/20 0.36
GPR35 Q9HC97 3/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9217742 0.90 NR4A1 (0.43) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL9041814 0.84 NR4A1 (0.51) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL9080057 0.84 ALDH1A1 (0.41) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL9039787 0.83 MPL (0.42) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL9077953 0.82 CNR2 (0.40) KDM4EALDH1A1HPGDHSD17B10NR4A1
SCHEMBL9079543 0.81 XDH (0.41) KDM4EALDH1A1HPGDHSD17B10NR4A1
SCHEMBL9077610 0.81 ALDH1A1 (0.44) ALDH1A1HPGDMEN1KMT2APTPN1
SCHEMBL9079015 0.77 KDM4E (0.51) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL9078240 0.77 KDM4E (0.50) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL4960266 0.76 KMT2A (0.44) KDM4EALDH1A1MEN1KMT2ADHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585382-A ANTICARCINOGENIC AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-17 US disclosed
US-5416089-A Antitumor agent THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-05-16 US disclosed
WO-1995000490-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-01-05 WO disclosed