SCHEMBL9040255

SCHEMBL9040255

COC(=O)C(=Cc1ccc(F)cc1)c1ccccc1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
CYP1A2 P05177 3/20 0.47
MEN1 O00255 2/20 0.47
CYP2C19 P33261 2/20 0.47
POLB P06746 2/20 0.47
TRPA1 O75762 2/20 0.46
MAPT P10636 4/20 0.46
ALDH1A1 P00352 3/20 0.46
CYP2C9 P11712 2/20 0.46
HPGD P15428 2/20 0.46
LMNA P02545 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CYP3A4 P08684 1/20 0.46
GAA P10253 1/20 0.46
ALOX12 P18054 1/20 0.46
NPC1 O15118 1/20 0.43
NFKB1 P19838 1/20 0.43
RAB9A P51151 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9078233 1.00 KMT2A (0.47) KMT2ACYP1A2MEN1CYP2C19POLB
SCHEMBL9148465 0.87 AKR1C3 (0.47) KMT2ACYP1A2MEN1CYP2C19POLB
SCHEMBL9040570 0.87 AKR1C3 (0.47) KMT2ACYP1A2MEN1CYP2C19POLB
SCHEMBL9039669 0.85 TRPA1 (0.49) POLBTRPA1MAPTALDH1A1NPC1
SCHEMBL9141932 0.85 TRPA1 (0.49) POLBTRPA1MAPTALDH1A1NPC1
SCHEMBL9143111 0.83 MAPT (0.43) KMT2AMEN1POLBTRPA1MAPT
SCHEMBL9040428 0.83 MAPT (0.43) KMT2AMEN1POLBTRPA1MAPT
SCHEMBL9037814 0.83 CYP1A2 (0.50) KMT2ACYP1A2MEN1CYP2C19POLB
SCHEMBL9078732 0.83 CYP1A2 (0.50) KMT2ACYP1A2MEN1CYP2C19POLB
SCHEMBL9141472 0.82 ALDH1A1 (0.46) KMT2AMEN1POLBTRPA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5585382-A ANTICARCINOGENIC AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-17 US disclosed
EP-0705250-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-04-10 EP disclosed
US-5416089-A Antitumor agent THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-05-16 US disclosed
WO-1995000490-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-01-05 WO disclosed