SCHEMBL904201

SCHEMBL904201

Cc1cc(C2=CCNCC2)cc(F)c1C

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 9/20 0.49
SIGMAR1 Q99720 2/20 0.47
QDPR P09417 3/20 0.45
HTR2A P28223 1/20 0.42
HTR7 P34969 1/20 0.42
HTR6 P50406 1/20 0.42
TGFBR1 P36897 1/20 0.40
ACVR1 Q04771 1/20 0.40
KCNH2 Q12809 1/20 0.40
CD274 Q9NZQ7 1/20 0.38
TLR9 Q9NR96 1/20 0.38
TLR7 Q9NYK1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4670817 0.81 SIGMAR1 (0.57) HTR2CSIGMAR1QDPRHTR2AHTR7
SCHEMBL16434840 0.81 HTR2C (0.57) HTR2CSIGMAR1QDPRHTR2AHTR7
Hydrochloric Acid SCHEMBL16422718 0.79 HTR2C (0.58) HTR2CSIGMAR1QDPRHTR2AHTR7
SCHEMBL10067587 0.78 QDPR (0.58) HTR2CSIGMAR1QDPR
SCHEMBL3386020 0.77 SIGMAR1 (0.59) HTR2CSIGMAR1QDPRHTR2AHTR7
Hydrochloric Acid SCHEMBL28669700 0.75 HTR2C (0.60) HTR2CSIGMAR1QDPRHTR2AHTR7
SCHEMBL5319444 0.75 SIGMAR1 (0.57) HTR2CSIGMAR1QDPRHTR2AHTR6
SCHEMBL14956908 0.75 QDPR (0.60) HTR2CSIGMAR1QDPRHTR7HTR6
SCHEMBL3383939 0.75 HTR2C (0.62) HTR2CSIGMAR1QDPRHTR2AHTR7
SCHEMBL5319876 0.74 SIGMAR1 (0.47) HTR2CSIGMAR1QDPRHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed