SCHEMBL9042091

SCHEMBL9042091

Cc1ccc(-n2cc(Br)cc2C#N)c(Br)c1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.37
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
ACHE P22303 1/20 0.31
OPRM1 P35372 1/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9040100 0.86 GABRB2 (0.35) ARACHE
SCHEMBL9041344 0.79 AR (0.33) AR
SCHEMBL9033966 0.79 ALDH1A1 (0.36) ARKMT2AMEN1
SCHEMBL9043599 0.78 LMNA (0.38) AROPRM1OPRK1
SCHEMBL9043916 0.73 POLB (0.35) AROPRM1OPRK1
SCHEMBL15561086 0.73 JAK2 (0.50) ARKMT2AMEN1
SCHEMBL9043421 0.73 KDM4E (0.36) ARKMT2A
SCHEMBL15561088 0.70 TSHR (0.35) AR
SCHEMBL15561129 0.68 KDM4E (0.40) ARKMT2AMEN1
SCHEMBL9041668 0.68 TSHR (0.31) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0480204-B1 Imidazole derivatives, potent and selective antagonists of angiotensin II receptor FUJISAWA PHARMACEUTICAL CO (JP) 1996-03-20 EP disclosed
US-5215994-A Treating or preventing hypertension or heart failure FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-06-01 US disclosed
US-5210092-A Hypotensive agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-11 US disclosed
EP-0480204-A1 Imidazole derivatives, potent and selective antagonists of angiotensin II receptor FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-15 EP disclosed