SCHEMBL9043285

SCHEMBL9043285

COc1ccc2[nH]c(-c3cccc(NC(C)=O)c3)nc2n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.61
KMT2A Q03164 5/20 0.61
ALDH1A1 P00352 4/20 0.61
MEN1 O00255 4/20 0.61
POLB P06746 4/20 0.61
TP53 P04637 3/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
HPGD P15428 2/20 0.61
HSD17B10 Q99714 2/20 0.61
DHODH Q02127 2/20 0.50
PARP1 P09874 1/20 0.50
COMT P21964 2/20 0.49
PIK3CA P42336 1/20 0.47
MTOR P42345 1/20 0.47
MAPT P10636 3/20 0.47
NPC1 O15118 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
FYN P06241 1/20 0.47
FAAH O00519 1/20 0.46
THRB P10828 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9043085 0.80 KDM4E (0.68) KDM4EKMT2AALDH1A1MEN1POLB
SCHEMBL9044486 0.80 KDM4E (0.71) KDM4EKMT2AALDH1A1MEN1POLB
SCHEMBL31661039 0.76 NPC1 (0.50) KDM4EALDH1A1TP53SMN1; SMN2HPGD
SCHEMBL2244254 0.76 KDM4E (1.00) KDM4EKMT2AALDH1A1MEN1POLB
SCHEMBL10875824 0.73 AURKA (0.47) KDM4EALDH1A1TP53SMN1; SMN2HPGD
SCHEMBL6125983 0.72 DGAT1 (0.53) KDM4EKMT2AALDH1A1MEN1SMN1; SMN2
SCHEMBL4057633 0.71 MEN1 (0.53) KDM4EKMT2AALDH1A1MEN1POLB
SCHEMBL24075063 0.70 KDM4E (0.69) KDM4EKMT2AALDH1A1MEN1POLB
SCHEMBL17280086 0.69 MAPT (0.60) KDM4EKMT2AALDH1A1MEN1POLB
SCHEMBL4053211 0.69 AURKA (0.62) KDM4EKMT2AALDH1A1MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700906-A1 Heterocyclic derivatives of N-phenylamides BRISTOL-MYERS SQUIBB COMPANY (US) 1996-03-13 EP disclosed
US-5496826-A ANTICONVULSANTS, MELATONERGIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1996-03-05 US disclosed