SCHEMBL9044486

SCHEMBL9044486

COc1ccc2[nH]c(-c3cccc(NC(C)=O)c3)nc2c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.71
KMT2A Q03164 8/20 0.71
MEN1 O00255 7/20 0.71
SMN1; SMN2 Q16637 6/20 0.71
ALDH1A1 P00352 5/20 0.71
POLB P06746 6/20 0.67
TP53 P04637 4/20 0.67
HPGD P15428 2/20 0.67
HSD17B10 Q99714 1/20 0.67
COMT P21964 2/20 0.66
MAPT P10636 6/20 0.62
NPC1 O15118 3/20 0.62
NPSR1 Q6W5P4 1/20 0.62
MMP2 P08253 2/20 0.60
MMP13 P45452 2/20 0.60
FYN P06241 1/20 0.55
RAB9A P51151 2/20 0.54
THRB P10828 1/20 0.54
RECQL P46063 1/20 0.54
ATM Q13315 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14302708 0.84 COMT (0.56) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL2244254 0.83 KDM4E (1.00) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL179157 0.81 NPC1 (0.63) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL9043285 0.80 KDM4E (0.61) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL12010985 0.78 COMT (0.83) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL9041717 0.78 STK33 (0.47) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL2740044 0.78 COMT (0.75) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL29349700 0.78 ALDH1A1 (0.72) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL20982455 0.78 ALDH1A1 (0.67) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL2324292 0.77 NPC1 (0.78) KDM4EKMT2AMEN1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700906-A1 Heterocyclic derivatives of N-phenylamides BRISTOL-MYERS SQUIBB COMPANY (US) 1996-03-13 EP disclosed
US-5496826-A ANTICONVULSANTS, MELATONERGIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1996-03-05 US disclosed