SCHEMBL9044286

SCHEMBL9044286

Nc1ccc(-n2cc(C(=O)O)c(=O)c3cc(F)c(N4CCNCC4)cc32)cc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.83
KDM4E B2RXH2 6/20 0.83
LMNA P02545 5/20 0.83
HSD17B10 Q99714 5/20 0.83
HPGD P15428 4/20 0.83
MEN1 O00255 1/20 0.66
KMT2A Q03164 1/20 0.66
TOP2A P11388 5/20 0.63
TOP2B Q02880 3/20 0.63
CYP1A2 P05177 1/20 0.63
CYP2C9 P11712 1/20 0.63
BRD4 O60885 1/20 0.63
TSHR P16473 1/20 0.63
HTT P42858 1/20 0.63
CYP2J2 P51589 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63
TOP1 P11387 2/20 0.57
POLB P06746 1/20 0.49
HSP90AA1 P07900 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sarafloxacin SCHEMBL311593 0.92 ALDH1A1 (0.98) ALDH1A1KDM4ELMNAHSD17B10HPGD
Sarafloxacin SCHEMBL379212 0.91 ALDH1A1 (1.00) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL9443539 0.91 ALDH1A1 (0.85) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL9443495 0.91 ALDH1A1 (0.85) ALDH1A1KDM4ELMNAHSD17B10HPGD
Sarafloxacin SCHEMBL23392485 0.90 ALDH1A1 (0.98) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL9443455 0.90 ALDH1A1 (0.83) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL11017466 0.90 ALDH1A1 (0.83) ALDH1A1KDM4ELMNAHSD17B10HPGD
Sarafloxacin SCHEMBL312072 0.90 ALDH1A1 (0.94) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL9443514 0.90 ALDH1A1 (0.83) ALDH1A1KDM4ELMNAHSD17B10HPGD
SCHEMBL9443467 0.88 ALDH1A1 (0.80) ALDH1A1KDM4ELMNAHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422485-B1 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1996-04-03 EP claimed
EP-0422485-B1 Quinolone carboxylic acid derivatives, process for their preparation and their use BAYER AG (DE) 1996-04-03 EP disclosed