SCHEMBL9044971

SCHEMBL9044971

COc1cccc(OCCC#N)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.56
MAOB P27338 6/20 0.50
MTNR1A P48039 1/20 0.50
MTNR1B P49286 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49
LMNA P02545 1/20 0.49
TSHR P16473 4/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
MEN1 O00255 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
RECQL P46063 1/20 0.48
KMT2A Q03164 1/20 0.48
ALOX15 P16050 1/20 0.48
HSD17B10 Q99714 1/20 0.48
APP P05067 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11764164 0.91 GAA (0.50) MAPK1MEN1KMT2A
Anisole SCHEMBL28263381 0.84 DRD2 (0.53) TSHRL3MBTL1MEN1CYP1A2CYP3A4
SCHEMBL1729519 0.82 MAPK1 (0.75) MAPK1MAOBMTNR1AMTNR1BNPSR1
SCHEMBL3728565 0.82 KMT2A (0.52) MAPK1NPSR1LMNAL3MBTL1KMT2A
SCHEMBL8195567 0.81 MAOB (0.53) MAPK1MAOBMTNR1AMTNR1BLMNA
SCHEMBL1810628 0.81 GAA (0.58) MAPK1MTNR1AMTNR1BNPSR1TSHR
SCHEMBL17361545 0.81 KDM4E (0.50) MAPK1MAOBLMNATSHRL3MBTL1
SCHEMBL18265518 0.81 GAA (0.42) CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL13684905 0.80 TBXAS1 (0.55)
SCHEMBL16502341 0.79 ALDH1A1 (0.54) MAPK1TSHRL3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749434-A1 BENZOTHIOPHENE, BENZOFURAN AND INDOLETHIAZEPINONES, OXAZEPINONES AND DIAZEPINONES AS INHIBITORS OF CELL ADHESION AND AS INHIBITORS OF HIV WARNER-LAMBERT COMPANY (US) 1996-12-27 EP disclosed
WO-1995024408-A1 BENZOTHIOPHENE, BENZOFURAN AND INDOLETHIAZEPINONES, OXAZEPINONES AND DIAZEPINONES AS INHIBITORS OF CELL ADHESION AND AS INHIBITORS OF HIV WARNER-LAMBERT COMPANY (US) 1995-09-14 WO disclosed
EP-0641792-A1 1,2-Dithiole derivatives and therapeutic agents containing them MITSUI TOATSU CHEMICALS, Inc. (JP) 1995-03-08 EP disclosed