SCHEMBL9045167

SCHEMBL9045167

COc1cccc2[nH]c(-c3ccccc3N)nc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.60
SMN1; SMN2 Q16637 4/20 0.59
ALDH1A1 P00352 4/20 0.59
HPGD P15428 3/20 0.59
HSD17B10 Q99714 2/20 0.59
CBFB Q13951 2/20 0.59
TP53 P04637 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
ALOX15 P16050 1/20 0.59
CYP2C19 P33261 1/20 0.59
GAA P10253 6/20 0.55
KDM4E B2RXH2 2/20 0.55
NPC1 O15118 2/20 0.55
MAPT P10636 2/20 0.55
RAB9A P51151 2/20 0.55
GLA P06280 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
SLC2A1 P11166 2/20 0.54
PDE5A O76074 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4563722 0.89 PARP1 (0.67) PARP1SMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL1170818 0.83 CBFB (0.69) PARP1SMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL9718865 0.82 GAA (0.65) PARP1SMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL29625822 0.79 HPSE (0.65) PARP1SMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL28027630 0.79 HPSE (0.65) PARP1SMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL14012670 0.78 MGAM (0.65) PARP1SMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL9044494 0.78 MGAM (0.71) PARP1SMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL8817550 0.77 PARP1 (0.63) PARP1SMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL9045175 0.77 ALDH1A1 (0.55) SMN1; SMN2ALDH1A1HPGDHSD17B10GAA
SCHEMBL4564339 0.77 PARP1 (0.63) PARP1SMN1; SMN2ALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700906-A1 Heterocyclic derivatives of N-phenylamides BRISTOL-MYERS SQUIBB COMPANY (US) 1996-03-13 EP disclosed
US-5496826-A ANTICONVULSANTS, MELATONERGIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1996-03-05 US disclosed