SCHEMBL9045281

SCHEMBL9045281

NC1CCN(c2c(F)cc3c(=O)c(C(=O)O)c[nH]c3c2-c2ccncc2F)C1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
TOP2A P11388 14/20 0.45
TOP2B Q02880 10/20 0.45
TOP1 P11387 4/20 0.43
RPS6KB1 P23443 1/20 0.43
MATK P42679 1/20 0.43
DYRK1A Q13627 1/20 0.43
MAPKAPK3 Q16644 1/20 0.43
PIM3 Q86V86 1/20 0.43
AURKB Q96GD4 1/20 0.43
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047491 1.00 ALDH1A1 (0.47) ALDH1A1POLBCHRM2CHRM1OPRM1
Hydrochloric Acid SCHEMBL9049612 0.99 ALDH1A1 (0.46) ALDH1A1POLBCHRM2CHRM1OPRM1
Hydrochloric Acid SCHEMBL9047371 0.84 TOP2A (0.42) ALDH1A1TOP2ATOP2BTOP1
SCHEMBL9047376 0.84 KDM4E (0.45) ALDH1A1POLBTOP2ATOP1KMT2A
SCHEMBL11013460 0.84 ALDH1A1 (0.53) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9046649 0.84 ALDH1A1 (0.47) ALDH1A1POLBCHRM2CHRM1OPRM1
Hydrochloric Acid SCHEMBL9044858 0.83 KDM4E (0.44) ALDH1A1POLBTOP2ATOP1KMT2A
SCHEMBL11015383 0.83 TOP1 (0.53) ALDH1A1POLBCHRM2CHRM1OPRM1
Hydrochloric Acid SCHEMBL9046844 0.83 ALDH1A1 (0.47) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9045950 0.79 KDM4E (0.41) ALDH1A1TOP2ATOP2BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713487-A1 NOVEL QUINOLONE CARBOXYLIC ACID DERIVATIVES DONG WHA PHARMACEUTICAL INDUSTRIAL CO. LTD. (KR) 1996-05-29 EP disclosed