SCHEMBL9045800

SCHEMBL9045800

CCc1cc2c(O)c(C(=O)OCC(C)C)cnc2s1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.46
ALDH1A1 P00352 7/20 0.43
HPGD P15428 3/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
TSHR P16473 1/20 0.41
P2RY12 Q9H244 1/20 0.40
KDM4E B2RXH2 4/20 0.39
HTT P42858 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP1A2 P05177 1/20 0.39
TMIGD3 P0DMS9 1/20 0.39
ADORA1 P30542 1/20 0.39
SELE P16581 1/20 0.38
VCAM1 P19320 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019066 0.89 NPSR1 (0.56) NPSR1ALDH1A1HPGDSMN1; SMN2KMT2A
SCHEMBL9044351 0.83 NPSR1 (0.46) NPSR1ALDH1A1HPGDSMN1; SMN2NPC1
SCHEMBL9046748 0.80 KDM4E (0.48) NPSR1ALDH1A1HPGDSMN1; SMN2NPC1
SCHEMBL6844296 0.80 NPSR1 (0.47) NPSR1ALDH1A1HPGDGAAMAPK1
SCHEMBL21708066 0.76 NPSR1 (0.43) NPSR1ALDH1A1HPGDMEN1GAA
SCHEMBL10998213 0.75 MAPT (0.46) ALDH1A1HPGDGAAMAPK1KDM4E
SCHEMBL5079627 0.73 ALDH1A1 (0.50) NPSR1ALDH1A1HPGDSMN1; SMN2NPC1
SCHEMBL7480184 0.73 GABRP (0.45) ALDH1A1HPGDGAAMAPK1KDM4E
SCHEMBL11579997 0.73 MAPT (0.44) ALDH1A1HPGDNPC1RAB9AMEN1
SCHEMBL11578876 0.73 MAPT (0.49) ALDH1A1HPGDMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0443568-B1 Fused thiophene derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-06-12 EP disclosed
US-5284661-A 4-Oxo-7-(biphenyl-4-yl)thieno(2,3-b)pyridines as antagonist of angiotensin II; hypertensive agents, cardiovascular disorders and strokes TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-02-08 US disclosed
EP-0443568-A1 Fused thiophene derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-08-28 EP disclosed