SCHEMBL9045900

SCHEMBL9045900

CN(CC1CCN(CCCCc2ccc(F)cc2)CC1)S(=O)(=O)c1cccc2cnccc12

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 1/20 0.47
P2RX7 Q99572 7/20 0.46
ROCK2 O75116 7/20 0.45
ROCK1 Q13464 7/20 0.45
HTR2A P28223 4/20 0.42
HTR7 P34969 4/20 0.42
HTR2C P28335 2/20 0.42
CCR2 P41597 1/20 0.42
HTR1A P08908 2/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
DRD2 P14416 1/20 0.41
HTR6 P50406 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9479252 0.99 FLT3 (0.47) FLT3P2RX7ROCK2ROCK1HTR2A
SCHEMBL9049718 0.88 P2RX7 (0.46) P2RX7ROCK2ROCK1HTR2AHTR7
Hydrochloric Acid SCHEMBL9478386 0.87 P2RX7 (0.46) P2RX7ROCK2ROCK1HTR2AHTR7
Hydrochloric Acid SCHEMBL9477834 0.87 HTR2A (0.45) FLT3P2RX7ROCK2ROCK1HTR2A
SCHEMBL9478929 0.86 HTR1A (0.48) P2RX7ROCK2ROCK1HTR2AHTR7
Hydrochloric Acid SCHEMBL9477785 0.84 ROCK2 (0.44) FLT3P2RX7ROCK2ROCK1HTR2A
Hydrochloric Acid SCHEMBL9480122 0.84 P2RX7 (0.44) P2RX7ROCK2ROCK1HTR2AHTR7
Hydrochloric Acid SCHEMBL9477689 0.83 P2RX7 (0.44) P2RX7ROCK2ROCK1
Hydrochloric Acid SCHEMBL9477303 0.83 P2RX7 (0.43) P2RX7ROCK2ROCK1HTR2AHTR7
SCHEMBL9046682 0.83 P2RX7 (0.45) P2RX7ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526342-B1 Isoquinolin-5yl-sulphonamides, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1996-12-04 EP claimed
US-5208243-A Analgesics ADIR ET COMPAGNIE (FR) 1993-05-04 US claimed