SCHEMBL9045967

SCHEMBL9045967

Nc1cc2c(O)n(CCc3ccc(F)cc3)cnc-2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 2/20 0.39
USP2 O75604 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
KDM5A P29375 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
HTT P42858 2/20 0.36
ALPL P05186 1/20 0.35
ALPG P10696 1/20 0.35
MGAT2 Q10469 1/20 0.33
MET P08581 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
MCHR1 Q99705 2/20 0.32
MITF O75030 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RAB9A P51151 1/20 0.32
ADORA2A P29274 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9048268 0.88 PSMB2 (0.39) SMN1; SMN2LMNAMAPTMAPK1HTT
SCHEMBL9046533 0.87 ADORA2A (0.44) HTTALDH1A1ADORA2A
SCHEMBL9471802 0.85 MAPK1 (0.45) SMN1; SMN2LMNAMAPTUSP2TSHR
SCHEMBL9047009 0.84 HSP90AA1 (0.43) MAPTHTTALDH1A1SLC5A1SLC5A2
SCHEMBL9046588 0.81 TAAR1 (0.35) ADORA2A
SCHEMBL9044408 0.80 KDM5A (0.43) KDM5AKDM5BHTTALPLALPG
SCHEMBL9045540 0.76 CSNK1D (0.42) LMNAKDM5AKDM5BMGAT2
SCHEMBL9342460 0.76 CDK9 (0.40) SMN1; SMN2LMNAMAPTHTTALDH1A1
SCHEMBL9053270 0.76 CNOT7 (0.42) SMN1; SMN2TSHRPTGS1PTGS2RAB9A
SCHEMBL9470878 0.74 CASR (0.38) SMN1; SMN2LMNAMAPTTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
US-5344932-A N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives TRUSTEES OF PRINCETON UNIVERSITY (US) 1994-09-06 US disclosed
US-5248775-A Pyrrolo(2,3-d)pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed