SCHEMBL9046142

SCHEMBL9046142

CNS(=O)(=O)Cc1ccc2[nH]cc(CCCNCCN(C)c3ncncc3OC)c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 9/20 0.54
HTR1D P28221 6/20 0.54
HTR1B P28222 6/20 0.54
HTR2A P28223 5/20 0.54
HTR2B P41595 2/20 0.54
HTR7 P34969 2/20 0.54
HTR5A P47898 2/20 0.54
HTR2C P28335 1/20 0.54
HTR1E P28566 1/20 0.54
HTR1F P30939 1/20 0.54
HTR3A P46098 1/20 0.54
SLC47A1 Q96FL8 1/20 0.54
SLC6A4 P31645 4/20 0.42
CYP1A2 P05177 4/20 0.38
CYP3A4 P08684 4/20 0.38
CYP2D6 P10635 4/20 0.38
CYP2C19 P33261 4/20 0.38
CYP2C9 P11712 3/20 0.38
HSD17B10 Q99714 2/20 0.38
USP2 O75604 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047164 0.90 HTR1D (0.54) HTR1AHTR1DHTR1BHTR2AHTR2B
SCHEMBL9047428 0.86 HTR1A (0.54) HTR1AHTR1DHTR1BHTR2AHTR2B
SCHEMBL9046137 0.85 HTR2A (0.49) HTR1AHTR1DHTR1BHTR2AHTR2B
Avitriptan SCHEMBL147315 0.77 HTR1D (0.55) HTR1AHTR1DHTR1BHTR2AHTR2B
Avitriptan SCHEMBL29633456 0.77 HTR1D (0.55) HTR1AHTR1DHTR1BHTR2AHTR2B
Avitriptan SCHEMBL4352074 0.76 HTR1D (0.54) HTR1AHTR1DHTR1BHTR2AHTR2B
SCHEMBL9047659 0.76 HTR1A (0.54) HTR1AHTR1DHTR1BHTR2AHTR2B
SCHEMBL9046688 0.75 HTR1D (0.49) HTR1AHTR1DHTR1BHTR2AHTR2B
SCHEMBL9045333 0.75 HTR1D (0.49) HTR1AHTR1DHTR1BHTR2AHTR2B
SCHEMBL9046625 0.74 HTR1A (0.49) HTR1AHTR1DHTR1BHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714896-A1 INDOL DERIVATIVES USEFUL FOR THE TREATMENT OF MIGRAINE, COMPOSITION AND UTILIZATION VITA-INVEST, S.A. (ES) 1996-06-05 EP claimed
EP-0714896-A1 INDOL DERIVATIVES USEFUL FOR THE TREATMENT OF MIGRAINE, COMPOSITION AND UTILIZATION VITA-INVEST, S.A. (ES) 1996-06-05 EP disclosed