Avitriptan

Avitriptan

SCHEMBL147315

CNS(=O)(=O)Cc1ccc2[nH]cc(CCCN3CCN(c4ncncc4OC)CC3)c2c1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 4/20 0.55
HTR1B P28222 4/20 0.55
HTR1A P08908 9/20 0.47
HTR7 P34969 2/20 0.47
SLC6A4 P31645 1/20 0.47
KCNH2 Q12809 1/20 0.47
HTR2A P28223 2/20 0.47
HTR2C P28335 1/20 0.47
HTR1E P28566 1/20 0.47
HTR1F P30939 1/20 0.47
HTR2B P41595 1/20 0.47
HTR3A P46098 1/20 0.47
HTR5A P47898 1/20 0.47
SLC47A1 Q96FL8 1/20 0.47
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Avitriptan SCHEMBL29633456 1.00 HTR1D (0.55) HTR1DHTR1BHTR1AHTR7SLC6A4
Avitriptan SCHEMBL4352074 0.99 HTR1D (0.54) HTR1DHTR1BHTR1AHTR7SLC6A4
SCHEMBL9045333 0.95 HTR1D (0.49) HTR1DHTR1BHTR1AHTR7SLC6A4
SCHEMBL4349219 0.91 HTR1A (0.49) HTR1AHTR7SLC6A4KCNH2ADRA2A
SCHEMBL6363083 0.91 HTR1A (0.49) HTR1AHTR7SLC6A4KCNH2ADRA2A
SCHEMBL4346029 0.90 HTR1A (0.48) HTR1DHTR1BHTR1AHTR7SLC6A4
SCHEMBL4345058 0.89 HTR1A (0.47) HTR1AHTR7SLC6A4KCNH2ADRA2A
Avitriptan SCHEMBL18396454 0.89 HTR1A (0.57) HTR1DHTR1BHTR1AHTR7SLC6A4
SCHEMBL6362007 0.88 HTR1D (0.51) HTR1DHTR1BHTR1AHTR7SLC6A4
Hydrochloric Acid SCHEMBL4349599 0.88 HTR1A (0.48) HTR1AHTR7SLC6A4KCNH2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1510 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4734974-A1 CANNABINOID COMPOSITION FOR USE IN THE TREATMENT OF PAIN AND/OR INFLAMMATION Mabewo Phytopharm AG (CH) 2026-05-06 EP claimed
WO-2026090164-A1 COMPOSITIONS COMPRISING ELISMETREP AND A SECOND THERAPEUTIC AGENT FOR TREATING OR PREVENTING MIGRAINE OR PAIN KALLYOPE, INC. (US) 2026-04-30 WO claimed
EP-4681714-A2 METHODS OF TREATING THE SYMPTOMS OF AUTISM SPECTRUM DISORDER MapLight Therapeutics, Inc. (US) 2026-01-21 EP claimed
US-12472255-B2 Pharmaceutical compositions comprising meloxicam AXSOME THERAPEUTICS, INC. (US) 2025-11-18 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
WO-2025003517-A1 CANNABINOID COMPOSITION FOR USE IN THE TREATMENT OF PAIN AND/OR INFLAMMATION MABEWO PHYTOPHARM AG (CH) 2025-01-02 WO claimed
EP-4483872-A1 CANNABINOID COMPOSITION FOR USE IN THE TREATMENT OF PAIN AND/OR INFLAMMATION Mabewo Phytopharm AG (CH) 2025-01-01 EP claimed
US-20240383973-A1 METHODS FOR TREATING CALCITONIN GENE-RELATED PEPTIDE (CGRP) - EXPRESSING CANCERS THE BOARD OF REGENTS OF THE UNIVERSITY OF OKLAHOMA (US) 2024-11-21 US claimed
US-20230391749-A1 CRYSTALLINE AND AMORPHOUS FORMS OF A DELTA-OPIOID MODULATOR TREVENA, INC. 2023-12-07 US claimed
EP-3999036-B1 ORODISPERSIBLE POWDER COMPOSITION COMPRISING A TRIPTAN BIOPHARMA SYNERGIES S L (ES) 2023-11-08 EP claimed
WO-2003015787-A1 USE OF BIBN4096 IN COMBINATION WITH OTHER ANTIMIGRAINE DRUGS FOR THE TREATMENT OF MIGRAINE BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-02-27 WO claimed
EP-1083918-A1 NOVEL THERAPEUTIC AGENTS THAT MODULATE 5-HT RECEPTORS Advanced Medicine, Inc. (US) 2001-03-21 EP claimed
WO-2001015677-A2 USE OF 5-HT1B/1D AGONISTS TO TREAT OTIC PAIN ALCON LABORATORIES, INC. (US) 2001-03-08 WO claimed
EP-0969842-A1 PHARMACEUTICAL COMPOSITION R.P. Scherer Limited (GB) 2000-01-12 EP claimed
WO-1999064044-A1 NOVEL THERAPEUTIC AGENTS THAT MODULATE 5-HT RECEPTORS ADVANCED MEDICINE, INC. (US) 1999-12-16 WO claimed
WO-1998042344-A1 PHARMACEUTICAL COMPOSITION R. P. SCHERER LIMITED (GB) 1998-10-01 WO claimed
US-5550239-A REACTING TRIALKYLSILYL N-PENTYLPIPERAZINYLPYRIMIDINE DERIVATIVE WITH 4-AMINO-3-IODO-BENZENESULFONAMIDE COMPOUND IN PALLADIUM CATALYZED HETEROANNULATION STEP, REMOVING TRIALKYLSILYL GROUP WITH MINERAL ACID, BASIFYING BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-27 US claimed
EP-0711769-A1 Improved process for large-scale production of BMS 180048 and analogs BRISTOL-MYERS SQUIBB COMPANY (US) 1996-05-15 EP claimed
US-5300506-A Indole-3-alkyl derivatives of alkoxypyrimidinylpiperazines BRISTOL-MYERS SQUIBB COMPANY (US) 1994-04-05 US claimed
EP-0548813-A1 Antimigraine 4-pyrimidinyl and pyridinyl derivatives of indol-3yl-alkyl piperazines Bristol-Myers Squibb Company (US) 1993-06-30 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12472255-B2 Pharmaceutical compositions comprising meloxicam CA9, CALCA, MC3R HTR1D 443/4885HTR1B 904/4885HTR1A 163/4885
US-20230391749-A1 CRYSTALLINE AND AMORPHOUS FORMS OF A DELTA-OPIOID MODULATOR OPRD1, OPRM1, OPRK1 HTR1D 368/4885HTR1B 556/4885HTR1A 545/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.