SCHEMBL9046569

SCHEMBL9046569

OCC#Cc1cccc(Oc2nccs2)c1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 1/20 0.44
TLR2 O60603 1/20 0.44
HAO1 Q9UJM8 9/20 0.43
ALOX5 P09917 5/20 0.41
ALDH1A1 P00352 1/20 0.36
MELK Q14680 1/20 0.36
EGFR P00533 1/20 0.35
P2RX3 P56373 1/20 0.35
ACACB O00763 1/20 0.34
ACACA Q13085 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9367822 0.82 TLR4 (0.47) TLR4TLR2HAO1ALOX5P2RX3
SCHEMBL2354820 0.76 TLR4 (0.49) TLR4TLR2ALOX5P2RX3
SCHEMBL9050229 0.76 TLR4 (0.42) TLR4TLR2HAO1ALOX5ALDH1A1
SCHEMBL9386945 0.75 ALOX5 (0.59) HAO1ALOX5ALDH1A1
SCHEMBL8052741 0.74 TLR4 (0.52) TLR4TLR2ALDH1A1P2RX3
SCHEMBL28888769 0.74 TLR4 (0.47) TLR4TLR2ALOX5P2RX3
SCHEMBL9051135 0.72 ALOX5 (0.39) HAO1ALOX5EGFR
SCHEMBL9045448 0.72 ALOX5 (0.68) ALOX5ACACBACACA
SCHEMBL12100240 0.71 TLR4 (0.52) TLR4TLR2P2RX3ACACBACACA
SCHEMBL8557561 0.71 TLR4 (0.52) TLR4TLR2ALDH1A1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0540673-B1 ACETYLENE DERIVATIVES HAVING LIPOXYGENASE INHIBITORY ACTIVITY ABBOTT LAB (US) 1996-10-16 EP disclosed
US-5559144-A LIPOXYGENASE INHIBITORS, INHIBITORS OF BIOSYNTHESIS OF LEUKOTRIENES ABBOTT LABORATORIES (US) 1996-09-24 US disclosed
US-5476873-A Inhibit biosynthesis of leukotrienes ABBOTT LABORATORIES (US) 1995-12-19 US disclosed