SCHEMBL9050229

SCHEMBL9050229

OCC#Cc1cccc(Oc2ccccn2)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 1/20 0.42
TLR2 O60603 1/20 0.42
ALOX5 P09917 1/20 0.42
HAO1 Q9UJM8 5/20 0.41
GRM5 P41594 2/20 0.41
ALDH1A1 P00352 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
FFAR1 O14842 1/20 0.39
PTGS2 P35354 2/20 0.39
LTA4H P09960 1/20 0.39
EGFR P00533 1/20 0.39
MAP4K4 O95819 1/20 0.39
IP6K1 Q92551 1/20 0.38
IP6K3 Q96PC2 1/20 0.38
IP6K2 Q9UHH9 1/20 0.38
MELK Q14680 1/20 0.38
SCN7A Q01118 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9368339 0.81 HAO1 (0.45) TLR4TLR2HAO1GRM5ALDH1A1
SCHEMBL9049445 0.81 TLR4 (0.47) TLR4TLR2HAO1GRM5FFAR4
SCHEMBL9386945 0.81 ALOX5 (0.59) ALOX5HAO1ALDH1A1FFAR1LTA4H
SCHEMBL9049379 0.80 ALOX5 (0.73) TLR4TLR2ALOX5HAO1GRM5
SCHEMBL9050814 0.80 GRM5 (0.47) HAO1GRM5
SCHEMBL9049679 0.80 L3MBTL1 (0.49) ALOX5HAO1ALDH1A1EGFRMAP4K4
SCHEMBL9049046 0.80 EGFR (0.43) ALOX5HAO1GRM5FFAR1EGFR
SCHEMBL29612417 0.77 TLR4 (0.56) TLR4TLR2GRM5ALDH1A1FFAR4
SCHEMBL12129555 0.77 TLR4 (0.56) TLR4TLR2GRM5ALDH1A1FFAR4
SCHEMBL9046569 0.76 TLR4 (0.44) TLR4TLR2ALOX5HAO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0540673-B1 ACETYLENE DERIVATIVES HAVING LIPOXYGENASE INHIBITORY ACTIVITY ABBOTT LAB (US) 1996-10-16 EP disclosed
US-5559144-A LIPOXYGENASE INHIBITORS, INHIBITORS OF BIOSYNTHESIS OF LEUKOTRIENES ABBOTT LABORATORIES (US) 1996-09-24 US disclosed
US-5476873-A Inhibit biosynthesis of leukotrienes ABBOTT LABORATORIES (US) 1995-12-19 US disclosed