SCHEMBL9047634

SCHEMBL9047634

C1=CCC2=c3nc(CCCN4CCCCC4)sc3=CC2=C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 11/20 0.35
DRD2 P14416 10/20 0.35
DRD4 P21917 8/20 0.35
HTR1A P08908 6/20 0.35
HTR7 P34969 6/20 0.35
HRH1 P35367 5/20 0.35
ADRA2A P08913 2/20 0.35
ADRA2C P18825 2/20 0.35
SLC6A2 P23975 2/20 0.35
ADRA1A P35348 2/20 0.35
HTR2B P41595 2/20 0.35
SIGMAR1 Q99720 2/20 0.35
HTR2A P28223 5/20 0.34
HTR2C P28335 3/20 0.34
DRD1 P21728 2/20 0.34
ADRA2B P18089 1/20 0.34
ADRA1D P25100 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
HTR1E P28566 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047746 0.94 L3MBTL1 (0.37) SIGMAR1HRH3L3MBTL1
Fumaric Acid SCHEMBL9050004 0.91 HRH3 (0.37) DRD3DRD2DRD4HTR1AHTR7
Fumaric Acid SCHEMBL9048779 0.82 HRH4 (0.37) DRD3DRD2DRD4HTR1AHTR7
SCHEMBL9048189 0.81
SCHEMBL9046288 0.77 SMN1; SMN2 (0.41) L3MBTL1
SCHEMBL9047118 0.76
SCHEMBL9098582 0.75 TBXAS1 (0.34)
SCHEMBL9045817 0.74
Fumaric Acid SCHEMBL9048442 0.73
SCHEMBL9097631 0.72 CYP2C9 (0.32) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749966-A1 5-HT 3 RECEPTOR AGONIST, NOVEL THIAZOLE DERIVATIVE, AND INTERMEDIATE THEREFOR YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-12-27 EP disclosed