SCHEMBL9047636

SCHEMBL9047636

CCOC(=O)c1cn(-c2ccon2)c2cc(F)c(F)c(N)c2c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.46
STAT3 P40763 2/20 0.44
KMT2A Q03164 2/20 0.39
TSHR P16473 1/20 0.36
CASP1 P29466 1/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 5/20 0.35
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 4/20 0.35
HSD17B10 Q99714 4/20 0.35
TBK1 Q9UHD2 1/20 0.35
P2RX7 Q99572 2/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 1/20 0.35
ROCK2 O75116 1/20 0.34
CDK1 P06493 1/20 0.34
PRKACA P17612 1/20 0.34
CDK2 P24941 1/20 0.34
CSNK1D P48730 1/20 0.34
GSK3A P49840 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045934 0.89 HTT (0.46) HTTSTAT3KMT2ATSHRCASP1
SCHEMBL9057013 0.85 HTT (0.46) HTTSTAT3KMT2ATSHRCASP1
SCHEMBL9045879 0.85 ALDH1A1 (0.40) HTTSTAT3KDM4EALDH1A1
SCHEMBL9046936 0.83 KMT2A (0.54) HTTSTAT3KMT2APKMHPGD
SCHEMBL9044625 0.83 HTT (0.41) HTTSTAT3KMT2ATSHRPKM
SCHEMBL9047198 0.81 STAT3 (0.59) HTTSTAT3KMT2APKMHPGD
SCHEMBL25069771 0.78 STAT3 (0.48) HTTSTAT3KMT2ATSHRCASP1
SCHEMBL9047236 0.78 STAT3 (0.60) HTTSTAT3KMT2ATSHRCASP1
SCHEMBL1243960 0.78 KMT2A (0.51) HTTSTAT3KMT2ATSHRHPGD
SCHEMBL9046444 0.77 STAT3 (0.51) HTTSTAT3KMT2AHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700912-A1 QUINOLONE DERIVATIVE OR SALT THEREOF, AND ANTIBACTERIAL CONTAINING THE SAME WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1996-03-13 EP disclosed