SCHEMBL9045879

SCHEMBL9045879

Nc1c(F)c(F)cc2c1c(=O)c(C(=O)O)cn2-c1ccon1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
HTT P42858 1/20 0.40
TOP1 P11387 1/20 0.39
GSK3B P49841 13/20 0.38
STAT3 P40763 1/20 0.38
FOXO1 Q12778 1/20 0.37
TOP2A P11388 1/20 0.35
TOP2B Q02880 1/20 0.35
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
HSP90AA1 P07900 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9044750 0.88 ALDH1A1 (0.41) ALDH1A1HTTTOP1GSK3BSTAT3
SCHEMBL9047564 0.87 ALDH1A1 (0.40) ALDH1A1HTTTOP1GSK3BSTAT3
SCHEMBL9047265 0.87 ALDH1A1 (0.40) ALDH1A1HTTTOP1GSK3BSTAT3
SCHEMBL9047636 0.85 HTT (0.46) ALDH1A1HTTSTAT3KDM4E
SCHEMBL9047248 0.83 ALDH1A1 (0.40) ALDH1A1HTTTOP1STAT3TOP2A
SCHEMBL9045282 0.81 LMNA (0.43) ALDH1A1HTTTOP1GSK3BTOP2A
SCHEMBL9045574 0.80 KCNH2 (0.38) ALDH1A1HTTTOP1GSK3BFOXO1
SCHEMBL9046944 0.76 ALDH1A1 (0.53) ALDH1A1HTTTOP1STAT3TOP2A
SCHEMBL9048884 0.75 GSK3B (0.35) GSK3BFOXO1POLB
SCHEMBL9048876 0.74 SLC2A1 (0.36) GSK3BFOXO1TOP2ATOP2BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700912-A1 QUINOLONE DERIVATIVE OR SALT THEREOF, AND ANTIBACTERIAL CONTAINING THE SAME WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1996-03-13 EP disclosed