SCHEMBL9048807

SCHEMBL9048807

O=C1C=C(O)CC(CCc2ccccc2F)(c2ccccc2)O1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.34
DAO P14920 2/20 0.34
OPRM1 P35372 2/20 0.33
OPRD1 P41143 2/20 0.33
OPRK1 P41145 2/20 0.33
TAAR1 Q96RJ0 1/20 0.33
MAOB P27338 1/20 0.33
NPC1 O15118 1/20 0.32
PAX8 Q06710 1/20 0.32
KLF5 Q13887 1/20 0.32
MPO P05164 2/20 0.32
DPP4 P27487 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
METAP2 P50579 1/20 0.32
LDHA P00338 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8007692 0.83 ALDH1A1 (0.38) EGFROPRM1MEN1KMT2ALDHA
SCHEMBL6604162 0.83 ALDH1A1 (0.38) EGFROPRM1MEN1KMT2ALDHA
SCHEMBL6606008 0.83 ASAH1 (0.37) EGFRMAOBNPC1ALDH1A1CYP2C9
SCHEMBL8008694 0.80 EGFR (0.35) EGFRTAAR1MEN1KMT2ALDHA
SCHEMBL8346206 0.80 EGFR (0.35) EGFRTAAR1MEN1KMT2ALDHA
SCHEMBL6175624 0.79 EGFR (0.38) EGFRLDHACYP1A2
SCHEMBL6605717 0.78 EGFR (0.38) EGFROPRM1NPC1KMT2ALDHA
SCHEMBL6302764 0.77 OPRM1 (0.35) DAOOPRM1OPRD1OPRK1TAAR1
SCHEMBL8341314 0.77 OPRK1 (0.39) OPRM1OPRD1OPRK1TAAR1
SCHEMBL8008514 0.77 OPRK1 (0.39) OPRM1OPRD1OPRK1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729464-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed