SCHEMBL9048810

SCHEMBL9048810

CS(=O)(=O)c1ccc(-n2cc(Cl)c(-c3ccc(Cl)cc3)n2)cc1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.63
KCNH2 Q12809 1/20 0.63
PTGS2 P35354 10/20 0.60
PTGS1 P23219 3/20 0.60
CA12 O43570 8/20 0.57
CA9 Q16790 8/20 0.57
CA1 P00915 3/20 0.55
CA2 P00918 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9048316 0.88 FAAH (0.61) FAAHKCNH2PTGS2PTGS1CA12
SCHEMBL9047622 0.86 FAAH (0.67) FAAHKCNH2PTGS2PTGS1CA12
SCHEMBL9048111 0.86 FAAH (0.60) FAAHKCNH2PTGS2PTGS1CA12
SCHEMBL9048935 0.84 PTGS2 (0.78) FAAHKCNH2PTGS2PTGS1CA12
SCHEMBL9047123 0.84 CA12 (0.80) FAAHKCNH2PTGS2PTGS1CA12
SCHEMBL23928634 0.84 CA12 (0.80) FAAHKCNH2PTGS2PTGS1CA12
SCHEMBL9048098 0.84 FAAH (0.58) FAAHKCNH2PTGS2PTGS1CA12
SCHEMBL9049345 0.83 FAAH (0.60) FAAHKCNH2PTGS2PTGS1CA12
SCHEMBL9047468 0.83 FAAH (0.57) FAAHKCNH2PTGS2PTGS1CA12
SCHEMBL9048763 0.83 FAAH (0.60) FAAHKCNH2PTGS2PTGS1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731796-A1 1,3,5-TRISUBSTITUTED PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP claimed
WO-1995015318-A1 1,3,5-TRISUBSTITUTED PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO claimed
EP-0731796-A1 1,3,5-TRISUBSTITUTED PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP disclosed
WO-1995015318-A1 1,3,5-TRISUBSTITUTED PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO disclosed