SCHEMBL9048935

SCHEMBL9048935

CS(=O)(=O)c1ccc(-n2cc(C=O)c(-c3ccc(Cl)cc3)n2)cc1

nearest known ligand 0.78

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.78
FAAH O00519 1/20 0.58
KCNH2 Q12809 1/20 0.58
CA12 O43570 7/20 0.55
CA9 Q16790 7/20 0.55
PTGS1 P23219 1/20 0.55
CA1 P00915 3/20 0.53
CA2 P00918 3/20 0.53
POLB P06746 1/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
NLRP3 Q96P20 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23928524 0.88 PTGS2 (0.78) PTGS2FAAHKCNH2CA12CA9
SCHEMBL23928490 0.87 PTGS2 (0.77) PTGS2CA12CA9POLBMEN1
SCHEMBL23928542 0.87 PTGS2 (0.66) PTGS2FAAHKCNH2CA12CA9
SCHEMBL23928584 0.86 PTGS2 (0.76) PTGS2CA12CA9CA1CA2
SCHEMBL23928623 0.84 PTGS2 (0.73) PTGS2FAAHKCNH2CA12CA9
SCHEMBL9048810 0.84 FAAH (0.63) PTGS2FAAHKCNH2CA12CA9
SCHEMBL9048316 0.83 FAAH (0.61) PTGS2FAAHKCNH2CA12CA9
SCHEMBL9047622 0.82 FAAH (0.67) PTGS2FAAHKCNH2CA12CA9
SCHEMBL9048111 0.82 FAAH (0.60) PTGS2FAAHKCNH2CA12CA9
SCHEMBL23928566 0.82 PTGS2 (0.69) PTGS2FAAHKCNH2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731796-A1 1,3,5-TRISUBSTITUTED PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP disclosed
WO-1995015318-A1 1,3,5-TRISUBSTITUTED PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO disclosed