SCHEMBL9049487

SCHEMBL9049487

COc1ccc2c(c1)C(=O)N(CCN1CCN(c3ccccc3OC)CC1)CO2

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 6/20 0.58
DRD2 P14416 6/20 0.58
DRD4 P21917 2/20 0.58
HTR7 P34969 2/20 0.52
DRD5 P21918 1/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
HTR1A P08908 3/20 0.52
ADRA1D P25100 2/20 0.52
ADRA1A P35348 2/20 0.52
ADRA1B P35368 2/20 0.52
ALDH1A1 P00352 2/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
ALOX12 P18054 1/20 0.52
HIF1A Q16665 1/20 0.52
HSD17B10 Q99714 1/20 0.52
KDM4E B2RXH2 2/20 0.51
TSHR P16473 1/20 0.51
GLA P06280 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9050903 0.90 DRD3 (0.52) DRD3DRD2DRD4HTR7DRD5
SCHEMBL9048438 0.89 ADRA1D (0.52) DRD3DRD2DRD4HTR7DRD5
SCHEMBL9050089 0.89 DRD3 (0.60) DRD3DRD2DRD4HTR7DRD5
SCHEMBL9050125 0.83 DRD3 (0.64) DRD3DRD2DRD4HTR7DRD5
SCHEMBL13448989 0.83 DRD2 (0.69) DRD3DRD2DRD4HTR7DRD5
SCHEMBL9047811 0.83 DRD3 (0.68) DRD3DRD2DRD4HTR7DRD5
SCHEMBL9049703 0.83 DRD3 (0.69) DRD3DRD2DRD4HTR7DRD5
SCHEMBL9047785 0.79 HTR2C (0.51) DRD3DRD2HTR7DRD5MEN1
SCHEMBL13448974 0.77 DRD2 (0.76) DRD3DRD2DRD4HTR7DRD5
SCHEMBL7470416 0.77 DRD2 (0.64) DRD3DRD2DRD4HTR7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0527081-B1 Substituted 3-piperazinylalkyl-2,3-dihydro-4H-1,3-benzoxazine-4-ones, their preparation and their therapeutical use PF MEDICAMENT (FR) 1996-01-03 EP claimed
US-5308844-A ANTIDEPRESSANT, ANXIOLYTIC AGENT, ANALGESIC, HYPOTENSIVE AGENT PIERRE FABRE MEDICAMENT (FR) 1994-05-03 US disclosed