SCHEMBL9049807

SCHEMBL9049807

COC(=O)Oc1c(C)csc1NC(=O)Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.56
POLB P06746 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C19 P33261 1/20 0.56
MAPK8 P45983 9/20 0.51
MAPK10 P53779 8/20 0.51
MAPK9 P45984 6/20 0.51
MAPT P10636 3/20 0.50
HPGD P15428 1/20 0.48
RAB9A P51151 2/20 0.45
ALDH1A1 P00352 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPC1 O15118 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
PDE4D Q08499 1/20 0.43
EPHX2 P34913 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1040586 0.80 MAPK8 (0.77) CYP1A2POLBCYP3A4CYP2C19MAPK8
SCHEMBL9052070 0.78 MAPT (0.54) CYP1A2POLBCYP3A4CYP2C19MAPK8
SCHEMBL9050785 0.74 MAPK8 (0.64) MAPK8MAPK10MAPK9MAPTHPGD
SCHEMBL9052092 0.72 KMT2A (0.51) CYP1A2POLBCYP3A4CYP2C19MAPK8
SCHEMBL23413572 0.69 NPC1 (0.76) CYP1A2POLBCYP3A4CYP2C19MAPK8
SCHEMBL13541545 0.69 HPGD (0.70) CYP1A2POLBCYP3A4CYP2C19MAPT
SCHEMBL12297957 0.68 ALDH1A1 (0.71) CYP1A2POLBCYP3A4CYP2C19MAPK8
SCHEMBL3712247 0.68 MAPK8 (0.78) CYP1A2POLBCYP3A4CYP2C19MAPK8
SCHEMBL11467089 0.67 MAPT (0.63) CYP1A2POLBCYP3A4CYP2C19MAPK8
SCHEMBL3714662 0.67 MAPK8 (0.80) MAPK8MAPK10MAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0717044-A1 Thienopyridone derivatives, their preparation and their use as NMDA-receptor antagonists MERCK PATENT GmbH (DE) 1996-06-19 EP disclosed