SCHEMBL9050477

SCHEMBL9050477

COc1ncnc(NCCN)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.46
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA7 P43166 2/20 0.38
CA13 Q8N1Q1 2/20 0.38
CHEK1 O14757 1/20 0.38
CHEK2 O96017 1/20 0.38
PDE5A O76074 2/20 0.36
LDHA P00338 1/20 0.35
FERMT2 Q96AC1 1/20 0.35
SYK P43405 1/20 0.34
LMNA P02545 2/20 0.34
HTT P42858 2/20 0.34
ENPP1 P22413 2/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 2/20 0.33
BRD4 O60885 1/20 0.33
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9046578 0.82 CYP1A2 (0.46) CYP1A2CYP2D6CHEK1CHEK2PDE5A
SCHEMBL8201557 0.74 ESR1 (0.49) ESR1CYP1A2CYP2D6LMNAHTT
SCHEMBL3817132 0.71 PDPK1 (0.45) ESR1CYP1A2PDE5ALMNAALDH1A1
SCHEMBL6701252 0.69 MAPK1 (0.66) LMNAHTTENPP1ALDH1A1MAPK1
SCHEMBL6233405 0.66 PDE5A (0.46) ESR1PDE5ALMNAEGFRMAPT
SCHEMBL12170630 0.66 GALR3 (0.40) PDE5ALDHALMNAHTTALDH1A1
SCHEMBL9049389 0.66 PDE1B (0.34) ESR1LMNAENPP1MAPK1SMN1; SMN2
SCHEMBL12170629 0.66 PDE5A (0.47) CYP1A2CHEK1PDE5ALMNAHTT
SCHEMBL17087808 0.65 ESR1 (0.56) ESR1ALDH1A1MAPK1EGFRMEN1
Hydrochloric Acid SCHEMBL898173 0.64 CYP1A2 (0.41) CYP1A2CYP2D6CHEK1CHEK2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714896-A1 INDOL DERIVATIVES USEFUL FOR THE TREATMENT OF MIGRAINE, COMPOSITION AND UTILIZATION VITA-INVEST, S.A. (ES) 1996-06-05 EP disclosed